29. Drouet, K. E.; Theodorakis, E. A. "Stereoselective Total Synthesis of Reveromycin B and C19-epi -Reveromycin B". Chemistry-A European J. 2000, 6, 1987-2001.PDF file, Supplement PDF

30. Drouet, K. E.; Ling, T.; Tran, H. V.; Theodorakis, E. A. "Enantioselective Synthesis of the [6,6] Spiroketal Core of Reveromycin A". Organic Lett. 2000, 2, 207-210. PDF file, Supplement PDF

31. Drouet, K. E.; Tran, H. V.; Theodorakis, E. A. "Efficient Synthesis of the C1-C8 Fragment of Reveromycins". Synthetic Commun. 2000, 30, 3617-3628. PDF file

32. Ling, T.; Kramer, B. A.; Palladino M. A.; Theodorakis, E. A. "Stereoselective Synthesis of (-) -Acanthoic Acid". Organic Lett. 2000, 2, 2073-2076. PDF file, Supplement PDF

33. Jamora, C.; Theodoraki, M.; Malhotra, V.; Theodorakis, E. A. "Investigation of the Biological Mode of Action of Clerocidin Using Whole Cell Assays". Bioorg. & Med. Chem. 2001, 9, 1365-1370. PDF file

34. Haidekker, M. A.; Ling, T.; Anglo, M.; Stevens, H.Y.; Frangos, J. A.; Theodorakis, E. A. "New Fluorescent Probes for the Measurement of Cell Membrane Viscosity". Chemistry & Biology 2001, 8, 123-131. PDF file

35. Lee, N.-J.; Kang, N.-I.; Cho, W..-J; Kim, S.-H.; Kang, K.-T.; Theodorakis, E. A. "Syntheses and Biological Activities of Medium Molecular Weights Polymers Containing Exo-3, 6-epoxy-1,2,3,6-tetrahydrophthalimidocaproic Acid". Polym. Int. 2001, 50, 1010-1015. PDF file

36. Ling, T.; Chowdhury, C.; Kramer, B. A.; Vong, B. G.; Palladino, M. A.; Theodorakis, E. A. "Enantioselective Synthesis of the Anti-inflammatory Agent (-)-Acanthoic Acid" J. Org. Chem. 2001, 66, 8843-8853. PDF file, Supplement PDF

37. Lee, N.-J.; Koo, J.-C.; Ju, S.-S.; Moon, S.-B.; Cho, W.-J.; Jeong, I.-C.; Lee, S.-J.; Cho, M.-Y.; Theodorakis, E. A. "Syntheses and Biological Activities of New Phthalimide-based Polymers Containing 5-Fluorouracil".Polym. Int. 2002, 51, 569-576. PDF file

38. Haidekker, M. A.; Tsai, A. G.; Brady, T.; Stevens, H. Y.; Frangos, J. A.; Theodorakis, E. A. "A Novel Approach to Blood Plasma Viscosity Measurement Using Fluorescent Molecular Rotors." Amer. J. Physiol. Heart Circ. Physiol. 2002, 282, H1609-H1614. PDF file

39. Ling, T.; Poupon, E.; Rueden, E. J.; Theodorakis, E. A. "Synthesis of (-) llimaquinone via a Radical Decarboxylation and Quinone Addition Reaction" Org. Lett. 2002, 4, 819-822. PDF file, Supplement PDF

40. Tisdale, E. J.; Chowdhury, C.; Vong, B. G.; Li, H.; Theodorakis, E. A. "Regioselective Synthesis of the Bridged Tricyclic Core of Garcinia Natural Products via Intramolecular Aryl Acrylate Cycloadditions"Org. Lett. 2002, 4, 909-912. PDF file, Supplement PDF

41. Haidekker, M. A.; Brady, T.; Wen, K.; Okada, C.; Stevens, H. Y.; Snell, J. M.; Frangos, J. A.; Theodorakis, E. A. "Phospholipid-bound Molecular Rotors: Synthesis and Characterization" Bioorg. & Med. Chem. 2002,10, 3627-3636. PDF file

42. Wen, K.; Chow, S.; Sanghvi, Y. S.; Theodorakis, E. A. "Synthesis of 2'-O-Methoxyethyl-Guanosine Using a Novel Silicon-Based Protecting Group" J. Org. Chem. 2002, 67. 7887-7889. PDF file, Supplement PDF

43. Ling, T.; Poupon, E.; Rueden, E. J.; Theodorakis, E. A. "Unified Synthesis of Quinone Sesquiterpenes Based on a Radical Decarboxylation and Quinone Addition Reaction" J. Am. Chem. Soc. 2002, 124, 12261-12267. PDF file, Supplement PDF

44. Ling, T.; Rivas, F.; Theodorakis, E. A. "Stereoselective Synthesis of the Fully Functionalized Core Fragment of Terpentecin" Tetrahedron Lett. 2002, 43, 9019-9022.
PDF file

45. Lee, N.-J.; Ju, S.-S.; Cho, W.-J.; Kim, S. H.; Kang, K.-T.; Brady, T.;Theodorakis, E. A. "Synthesis and Antitumor Activity of Medium MolecularWeight Phthalimide-Polymers of Camptothecin" Eur. Polymer J. 2003, 39, 367-374. PDF file

46. Lee, N.-J.; Theodorakis, E. A. "Synthesis and Antitumor Activity of Phthalimide-Based Polymers Containing Camptothecin" Macromol. Res. 2003, 11, 47-52. PDF file

47. Tisdale, E. J.; Kochman, D. A.; Theodorakis, E. A. "Total Synthesis of Atroviridin" Tetrahedron Lett. 2003, 44, 3281-3284. PDF file

48. Chow, S.; Wen, K.; Sanghvi, Y. S.; Theodorakis, E. A. "Novel Synthesis of 2'-O-Methylguanosine" Bioorg. & Med. Chem. Lett. 2003, 13, 1631-1634. PDF file

49. Tisdale, E. J.; Li, H.; Vong, B. G.; Kim, S. H.; Theodorakis, E. A. "Regioselective Synthesis of the Tricyclic Core of Lateriflorone" Org. Lett. 2003, 5, 1491-1494.
PDF file, Supplement PDF

50. Vong, B. G.; Abraham, S.; Xiang, A. X.; Theodorakis, E. A. "Synthetic Studies on Borrelidin; Enantioselective Synthesis of the C1-C12 Fragment" Org. Lett. 2003, 5, 1617-1620. PDF file, Supplement PDF

51. Lee, N.-J.; Ju, S.-S.; Cho, W.-J.; Kim, S. H.; Kang, K.-T.; Brady, T.; Theodorakis, E. A. "Synthesis and Antitumor Activity of Medium Molecular Weight Phthalimide-Polymers of Camptothecin" Polym. Int. 2003, 52, 1339-1345. PDF file

52. Tisdale, E. J.; Vong, B. G.; Li, H.; Kim, S. H.; Chowdhury, C.; Theodorakis, E. A. "Total Synthesis of Seco-lateriflorone" Tetrahedron 2003, 59, 6873-6887. PDF file

53. Lam, T.; Ling, T.; Chowdhury, C.; Chao, T.-H.; Bahjat, F. R.; Lloyd, G. K.; Moldawer, L. L.; Palladino, M. A.; Theodorakis, E. A. "Synthesis of a Novel Family of Diterpenes and their Evaluation as Anti-inflammatory Agents" Bioorg. & Med. Chem. Lett. 2003, 13, 3217-3221. PDF file

54. Palladino, M. A.; Bahjat, F. R.; Theodorakis, E. A.; Moldawer, L. L. "Anti TNF-a Therapies: The Next Generation" Nature Reviews Drug Discovery 2003, 2, 736-746. PDF file

55. Chow, S.; Wen, K.; Sanghvi, Y. S.; Theodorakis, E. A. "MDPSCl2: A New Protecting Group for Chemoselective Synthesis of 2'-O-Alkylated Guanosines" Nucleos. Nucleot. Nucl. Acids 2003, 22, 583-587. PDF file

56. Tisdale, E. J.; Slobodov, I; Theodorakis, E. A. "Biomimetic Total Synthesis of Forbesione and Desoxymorellin Utilizing a Tandem Claisen/Diels-Alder/Claisen Rearrangement" Org. Biomol. Chem. 2003, 1, 4418-4422. PDF file, Supplement PDF

57. Brady, T.; Kim, S.; Wen, K.; Theodorakis, E. A. "Stereoselective Total Synthesis of (+)-Norrisolide" Angew. Chem. Int. Ed. 2004, 43, 739-742. PDF file, Supplement PDF

58. Oka, N.; Sanghvi, Y. S.; Theodorakis, E. A. "1,2-Ethylene-3,3-Bis(4'-4"-Dimethoxytrityl Chloride) (E-DMT): Synthesis and Applications of a Novel Protecting Reagent" Synlett 2004, 5, 823-826. PDF file

59. Kim, C.; Brady, T.; Kim, S.; Theodorakis, E. A. "Synthesis of Fused Tetrahydrofuran-≥-lactone Motifs via a One-Pot Ring Expansion of Cyclopropane Rings" Synth. Commun. 2004, 34, 1951-1965. PDF file

60. Ghosh, S.; Rivas, F.; Fischer, D.; Gonzalez, M. A. "Stereoselective Synthesis of the ABC Ring System of Norzoanthamine" Org. Lett. 2004, 6, 941-944. PDF file, Supplement PDF

61. Lee, N.-J.; Lee, S.-J.; Kim, S.-H.; Soo, K.-Y.; Moon, S.-B.; Kang, K.-T.; Theodorakis, E. A. "Synthesis and in vitro Antitumour Activity of Phthalimide-Based Polymers Containing Camptothecin" Eur. Polymer J. 2004, 40, 1291-1296. PDF file

62. Oka, N.; Sanghvi, Y. S.; Theodorakis, E. A. "3,3'-Oxybis(Dimethoxytrityl Chloride) (O-DMT): Synthesis and Applications of a Novel Bifunctional Protecting Group" Bioorg. & Med. Chem. 2004, 14, 3241-3244. PDF file

63. Haidekker, M. A.; Brady, T. P.; Chalian, S. H.; Akers, W.; Lichlyter, D.; Theodorakis, E. A. "Hydrophilic Molecular Rotor Derivatives: Synthesis and Characterization" Bioorg. Chem. 2004, 32, 274-289. PDF file

64. Gonzalez, M. A.; Ghosh, S.; Rivas, F.; Fischer, D.; Theodorakis, E. A. "Synthesis of (+)- and (-)-Isocarvone" Tetrahedron Lett. 2004, 45, 5039-5041. PDF file

65. Theodorakis, E. A.; Ling, T.; Rueden, E. J.; Poupon E.; Kim S. H. "Quinone Sesquiterpenes: A Challenge for the Development of a New Synthetic Methodology" Strategies and Tactics in Organic Synthesis, 2004, Vol. 5, 111-131. PDF file

66. Vong, B. G.; Kim, S. H.; Abraham, S.; Theodorakis, E. A. "Stereoselective Total Synthesis of
(-)-Borrelidin" Angew. Chem. Int. Ed. 2004, 43, 3947-3951. PDF file, Supplement PDF

67. Tisdale, E. J.; Slobodov, I; Theodorakis, E. A. "Unified Synthesis of Caged Garcinia Natural Products Based on a Site-Selective Claisen/Diels-Alder/Claisen Rearrangement" Proc. Nat. Acad. Sci. USA 2004, 101, 12030-12035. PDF file, Supplement PDF

68. Brady, T. P.; Wallace, E. K.; Kim, S. H.; Guizunnti, G.; Malhotra, V.; Theodorakis, E. A. "Fragmentation of Golgi Membranes by Norrisolide and Designed Analogues" Bioorg. & Med. Chem. Lett. 2004, 14, 5035-5039. PDF file

 

 
 
 
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