make your own website



154. "Chiral resolution of a caged xanthone and evaluation across a broad spectrum of breast cancer subtypes" Chantarasriwong, O.; Dorwart, T. J.; Morales, T. H.; Maggio, S. F.; Settle, A. L.; Milcarek, A. T.; Alpaugh, M. L.; Theodoraki, M. A.; Theodorakis, E. A. Bioorg. Chem. 2019 93, 103303.

153. "Synthesis, structure-activity relationship and in vitro pharmacodynamics of A-ring modified caged xanthones in a preclinical model of inflammatory breast cancer" Chantarasriwong, Oraphin; Milcarek, Andrew T.; Morales, Theodore H.; Settle, Aspen L.; Rezende, Celso O.; Althufairi, Bashayer D.; Theodoraki, Maria A.; Alpaugh, Mary L.; Theodorakis. Emmanuel A.; Milcarek, Andrew T. European Journal of Medicinal Chemistry, 2019, 168(15), 405-413. 

152. "Marine Spirotetronates: Biosynthetic Edifices That Inspire Drug Discovery" Braddock, Alexander A.; Theodorakis, Emmanuel A. Marine Drugs, 2019, 17(4), 232. 

151. "Solvation-guided design of fluorescent probes for discrimination of amyloids" Cao, K. J.; Elbel, K. M.; Cifelli, J. L.; Cicera, J.; Sigurdson, C. J.; Paesani, F.; Theodorakis, E. A.; Yang, J. Scientific Reports, 2018, 8, 6950. 

150. "Caged Garcinia Xanthones: Synthetic Studies and Pharmacophore Evaluation" Chantarasriwong, Oraphin; Althufairi, Bashayer D.; Checchia, Nicholas J.; Theodorakis, Emmanuel A. Studies in Natural Products Chemistry, 2018, 58, 93-131. 

149. "Caged Garcinia Xanthones, a Novel Chemical Scaffold with Potent Antimalarial Activity" Ke, Hangjun; Morrisey, Joanne M.; Qu, Shiwei; Chantarasriwong, Oraphin; Mather, Michael W.; Theodorakis, Emmanuel A. Antimicrobial Agents and Chemotherapy, 2017, 61(1), e01220-16. 

148. "Gambogic acid identifies an isoform-specific druggable pocket in the middle domain of Hsp90β" KYim, Kendrick H.; Prince, Thomas L.; Qu, Shiwei; Bai, Fang; Jennings, Patricia A.; Onuchic, José N.; Theodorakis, Emmanuel A. PNAS, 2016, 113, (33), E4801-E4809. 

147. "Ratiometric mechanosensitive fluorescent dyes: design and applications" Haidekker, Mark A.; Theodorakis, Emmanuel A. J. Mater. Chem. C, 2016, 4, 2707-2718. 

146. "Spontaneously-forming spheroids as an in vitro cancer cell model for anticancer drug screening" Theodoraki, Maria A.; Rezende Jr, Celso O.; Chantarasriwong, Oraphin; Corben, Adriana D. Theodorakis, Emmanuel A. Alpaugh, Mary L. J. Mater. Oncotarget, 2015, 6(25), 21255–21267. 

145. "Total Synthesis and Structural Revision of Antibiotic CJ‐16,264" Nicolaou, K.C.; Shah, Akshay A.; Korman, Henry; Khan, Tabrez; Shi, Lei; Worawalai, Wisuttaya; Theodorakis, Emmanuel A. Angew. Chem. Int. Ed., 2015, 54, 9203-9208. 

144. "Real-Time Monitoring of Alzheimer’s-Related Amyloid Aggregation via Probe Enhancement–Fluorescence Correlation Spectroscopy" Guan, Yinghua; Cao, Kevin J.; Cantlon, Adam; Elbel, Kristyna; Theodorakis, Emmanuel A.; Walsh, Dominic M.; Yang, Jerry; Shah, Jagesh V. ACS Chem. Neurosci., 2015, 6, 9, 1503-1508.

143. "Spirotetronate Polyketides as Leads in Drug Discovery" GLacoske, Michelle H.; Theodorakis, Emmanuel A. J. Nat. Prod. 2015, 78 (3), 562-575. 

142. "The Fe-S cluster-containing NEET proteins mitoNEET and NAF-1 as chemotherapeutic targets in breast cancer" Bai, Fang; Morcos, Faruck; Sohn, Yang-Sung; Darash-Yahana, Merav; Rezende, Celso O.; Lipper, Colin H.; Paddock, Mark L; Song, Luhua; Luo, Yuting; Holt, Sarah H.; Tamir, Sagi; Theodorakis, Emmanuel A. Jennings, Patricia A.; Onuchic, José N.; Mittler, Ron; Nechushtai, Rachel. PNAS, 2015, 112(12), 3698-3703.

141. "Synthetic Strategies Toward the Decalin Motif of Maklamicin and Related Spirotetronates" Lacoske Michelle H.; Xu, Jing; Mansour, Noel; Gao, Chao; Theodorakis, Emmanuel A. Org Chem Front., 2015, 2(4), 388–393. 

140. "3, 4-diaminobenzoic acid derivatives as inhibitors of the oxytocinase subfamily of M1 aminopeptidases with immune-regulating properties" Papakyriakou, Athanasios; Zervoudi, Efthalia; Tsoukalidou, Sofia; Mauvais, Francois-Xavier; Sfyroera, Georgia; Mastellos, Dimitrios C.; Endert, Peter Van; Theodorakis, Emmanuel A.; Vourloumis, Dionisios; Stratikos, Efstratios. J. Med. Chem., 2015, 58, 3, 1524-1543. 

139. "Cyclopenta [b] naphthalene cyanoacrylate dyes: synthesis and evaluation as fluorescent molecular rotors" Kocsis, Laura S.; Elbel, Kristyna M.; Hardigree, Billie A.; Brummond, Kay M.; Haidekker, Mark A.; Theodorakis, Emmanuel A. Org. Biomol. Chem., 2015, 13, 2965-2973. 

138. “Apparent shear sensitivity of molecular rotors in various solvents” Mustafic, A.; Elbel, K. M.; Theodorakis, E. A.; Haidekker, M. J. Fluoresc. 2015, 25, 729-738.